SCHEMBL28514928

SCHEMBL28514928

COc1cc(B2OC(C)(C)C(C)(C)O2)cc(OC)c1N1CCN(C)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 3/20 0.39
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
HRH4 Q9H3N8 1/20 0.36
ACHE P22303 1/20 0.35
BACE1 P56817 1/20 0.35
SIRT6 Q8N6T7 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
CSF1R P07333 1/20 0.34
MAOA P21397 2/20 0.33
MAOB P27338 2/20 0.33
SLC6A4 P31645 1/20 0.33
CCNT1 O60563 1/20 0.32
CDK4 P11802 1/20 0.32
CCNA2 P20248 1/20 0.32
CCND1 P24385 1/20 0.32
CDK2 P24941 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
CCNH P51946 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28504440 0.92 CCR4 (0.39) CCR4DRD2DRD3HRH4ACHE
SCHEMBL28502430 0.91 CCR4 (0.36) CCR4DRD2DRD3HRH4ACHE
SCHEMBL28504451 0.88 ALDH1A1 (0.36) CCR4SMN1; SMN2
SCHEMBL2798649 0.82 DRD2 (0.49) DRD2DRD3ACHECSF1RMAOB
SCHEMBL24723411 0.81 LPL (0.33) CCR4HRH4ACHESMN1; SMN2
SCHEMBL19099105 0.81 MEN1 (0.38) SMN1; SMN2CSF1RMAOAMAOBSLC6A4
SCHEMBL2802127 0.80 DRD2 (0.49) DRD2DRD3CSF1R
SCHEMBL28499596 0.79 ROCK1 (0.39) HRH4SMN1; SMN2
SCHEMBL24722850 0.78 CCR4 (0.37) CCR4HRH4SMN1; SMN2
SCHEMBL24722841 0.76 HRH4 (0.35) DRD2DRD3HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed