SCHEMBL2850486

SCHEMBL2850486

CCCc1c(OC(=O)NCCc2ccncc2)cnn1-c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
KDM4E B2RXH2 1/20 0.44
TAAR1 Q96RJ0 1/20 0.42
LMNA P02545 2/20 0.42
PKM P14618 1/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPK14 Q16539 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ABCB1 P08183 2/20 0.37
MAPK1 P28482 2/20 0.37
GAA P10253 1/20 0.37
SMO Q99835 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856900 0.94 MAPT (0.47) MAPTTAAR1LMNAPKMMAPK14
SCHEMBL2860461 0.91 TAAR1 (0.54) MAPTTAAR1LMNAPKMABCB1
SCHEMBL2848346 0.89 MAPT (0.55) MAPTTAAR1LMNAPKMRAB9A
SCHEMBL2857882 0.89 MAPT (0.43) MAPTTAAR1LMNAPKMKMT2A
SCHEMBL2856513 0.89 TAAR1 (0.51) MAPTTAAR1LMNAPKMKMT2A
SCHEMBL2850361 0.87 ABCB1 (0.48) MAPTTAAR1LMNAPKMMEN1
SCHEMBL2858349 0.87 CNR1 (0.44) MAPTTAAR1LMNAPKMMAPK14
SCHEMBL2855564 0.86 CNR1 (0.48) MAPTTAAR1LMNAPKMMAPK14
SCHEMBL2855797 0.86 CNR1 (0.47) MAPTTAAR1LMNAPKMMAPK14
SCHEMBL2857965 0.85 TAAR1 (0.47) MAPTTAAR1LMNAPKMABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed