SCHEMBL28507129

SCHEMBL28507129

Cc1cc(-c2cnc3[nH]cc(-c4ccc(CO)cc4)c3c2)cc(C)c1N1CCN(C)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 9/20 0.59
MAP3K11 Q16584 7/20 0.57
MAP4K1 Q92918 6/20 0.57
IKBKB O14920 2/20 0.53
CHUK O15111 2/20 0.53
ABL1 P00519 2/20 0.53
INSR P06213 2/20 0.53
CDK2 P24941 2/20 0.53
FLT3 P36888 2/20 0.53
IL2 P60568 3/20 0.52
SGK1 O00141 1/20 0.52
AURKA O14965 1/20 0.52
PRKAB2 O43741 1/20 0.52
ROCK2 O75116 1/20 0.52
NTRK1 P04629 1/20 0.52
LCK P06239 1/20 0.52
CDK1 P06493 1/20 0.52
IGF1R P08069 1/20 0.52
MET P08581 1/20 0.52
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513938 0.88 MAP4K1 (0.56) TNIKMAP3K11MAP4K1IKBKBCHUK
SCHEMBL21592630 0.87 NTRK1 (0.58) TNIKMAP3K11MAP4K1IL2NTRK1
SCHEMBL28517248 0.86 MAP4K1 (0.64) TNIKMAP3K11MAP4K1IL2SGK1
SCHEMBL28503427 0.86 MAP4K1 (0.54) TNIKMAP3K11MAP4K1IKBKBCHUK
SCHEMBL28510217 0.85 MAP4K1 (0.56) TNIKMAP3K11MAP4K1IKBKBCHUK
SCHEMBL21592774 0.85 MAP4K1 (0.71) TNIKMAP3K11MAP4K1IL2SGK1
SCHEMBL28499799 0.85 SGK1 (0.63) TNIKMAP3K11MAP4K1IL2SGK1
SCHEMBL28906168 0.84 MAP4K1 (0.56) TNIKMAP3K11MAP4K1IL2SGK1
SCHEMBL21592566 0.84 MAP4K1 (0.65) TNIKMAP3K11MAP4K1IL2SGK1
SCHEMBL21592582 0.83 TNIK (0.54) TNIKMAP3K11MAP4K1IL2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed