SCHEMBL28507697

SCHEMBL28507697

CN1CCN(c2ccc(-c3cnc4c(c3)c(I)cn4C(=O)OC(C)(C)C)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.48
MAP4K1 Q92918 15/20 0.45
IL2 P60568 1/20 0.45
LCK P06239 1/20 0.44
MAP4K3 Q8IVH8 1/20 0.44
FYN P06241 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28506162 0.88 CHEK1 (0.48) CHEK1MAP4K1IL2LCKMAP4K3
SCHEMBL28502006 0.88 MAP4K1 (0.44) CHEK1MAP4K1IL2
SCHEMBL28514984 0.87 FGFR1 (0.38) CHEK1MAP4K1LCKMAP4K3
SCHEMBL22971783 0.86 MAP3K11 (0.51) MAP4K1LCK
SCHEMBL21590168 0.85 WDR5 (0.41) CHEK1MAP4K1
SCHEMBL28506918 0.84 MAP4K1 (0.39) MAP4K1IL2LCKMAP4K3FYN
SCHEMBL21590350 0.83 CHEK1 (0.45) CHEK1MAP4K1IL2LCKMAP4K3
SCHEMBL31553241 0.83 PAK1 (0.46) MAP4K1
SCHEMBL28499816 0.82 NR1H2 (0.43)
SCHEMBL719094 0.80 GSK3B (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed