SCHEMBL28508649

SCHEMBL28508649

Cc1cc(Cl)ccc1N1CCC[C@@H](N(C)C(=O)OC(C)(C)C)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.42
DDR1 Q08345 3/20 0.41
RET P07949 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
KIF18A Q8NI77 1/20 0.39
PDE10A Q9Y233 1/20 0.39
KDM4D Q6B0I6 1/20 0.38
PROKR1 Q8TCW9 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD11B1 P28845 1/20 0.38
GRM5 P41594 1/20 0.38
PPARA Q07869 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
BTK Q06187 2/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28506403 1.00 AKR1C3 (0.42) AKR1C3DDR1RETHRH3KIF18A
SCHEMBL28506133 0.94 PDE10A (0.43) AKR1C3DDR1HRH3PDE10AKDM4D
SCHEMBL28508706 0.94 PDE10A (0.43) AKR1C3DDR1HRH3PDE10AKDM4D
SCHEMBL27128619 0.89 DDR1 (0.41) DDR1RETKIF18APDE10AKDM4D
SCHEMBL27128597 0.89 NPC1 (0.42) DDR1RETKIF18APDE10AKDM4D
SCHEMBL27139761 0.89 DDR1 (0.41) DDR1RETKIF18APDE10AKDM4D
SCHEMBL28504211 0.88 AKR1C3 (0.46) AKR1C3DDR1PDE10AKDM4DLMNA
SCHEMBL24628490 0.82 PDE10A (0.45) DDR1PDE10AKDM4DHSD11B1GRM5
SCHEMBL29772858 0.82 PDE10A (0.45) DDR1PDE10AKDM4DHSD11B1GRM5
SCHEMBL29772884 0.82 PDE10A (0.45) DDR1PDE10AKDM4DHSD11B1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed