SCHEMBL28508706

SCHEMBL28508706

Cc1cc(Cl)ccc1N1CC[C@H](N(C)C(=O)OC(C)(C)C)C1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.43
AKR1C3 P42330 1/20 0.43
AAK1 Q2M2I8 1/20 0.42
HSD11B1 P28845 1/20 0.41
NOTUM Q6P988 2/20 0.41
KDM4D Q6B0I6 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
DDR1 Q08345 4/20 0.40
GRM5 P41594 1/20 0.39
PIK3CD O00329 1/20 0.39
MCHR1 Q99705 1/20 0.38
USP30 Q70CQ3 3/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28506133 1.00 PDE10A (0.43) PDE10AAKR1C3AAK1HSD11B1NOTUM
SCHEMBL28504211 0.94 AKR1C3 (0.46) PDE10AAKR1C3AAK1HSD11B1NOTUM
SCHEMBL28506403 0.94 AKR1C3 (0.42) PDE10AAKR1C3AAK1HSD11B1KDM4D
SCHEMBL28508649 0.94 AKR1C3 (0.42) PDE10AAKR1C3AAK1HSD11B1KDM4D
SCHEMBL24628490 0.88 PDE10A (0.45) PDE10AAAK1HSD11B1NOTUMKDM4D
SCHEMBL29772858 0.88 PDE10A (0.45) PDE10AAAK1HSD11B1NOTUMKDM4D
SCHEMBL29772884 0.88 PDE10A (0.45) PDE10AAAK1HSD11B1NOTUMKDM4D
SCHEMBL27128619 0.82 DDR1 (0.41) PDE10AAAK1HSD11B1NOTUMKDM4D
SCHEMBL27128597 0.82 NPC1 (0.42) PDE10AAAK1HSD11B1NOTUMKDM4D
SCHEMBL27139761 0.82 DDR1 (0.41) PDE10AAAK1HSD11B1NOTUMKDM4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed