SCHEMBL24628490

SCHEMBL24628490

CN(C(=O)OC(C)(C)C)C1CCN(c2ccc(Cl)cc2F)C1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.45
FPR1 P21462 2/20 0.43
FPR2 P25090 2/20 0.43
USP30 Q70CQ3 1/20 0.43
AAK1 Q2M2I8 1/20 0.42
DDR1 Q08345 4/20 0.41
PDK2 Q15119 2/20 0.41
HSD11B1 P28845 1/20 0.41
KDM4D Q6B0I6 2/20 0.41
NOTUM Q6P988 1/20 0.40
MAPT P10636 1/20 0.38
GRM5 P41594 1/20 0.38
CCR4 P51679 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP3A5 P20815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29772884 1.00 PDE10A (0.45) PDE10AFPR1FPR2USP30AAK1
SCHEMBL29772858 1.00 PDE10A (0.45) PDE10AFPR1FPR2USP30AAK1
SCHEMBL28508706 0.88 PDE10A (0.43) PDE10AUSP30AAK1DDR1HSD11B1
SCHEMBL28506133 0.88 PDE10A (0.43) PDE10AUSP30AAK1DDR1HSD11B1
SCHEMBL4288048 0.87 PDE10A (0.43) PDE10AFPR1FPR2USP30AAK1
SCHEMBL31485219 0.87 PDE10A (0.43) PDE10AFPR1FPR2USP30AAK1
SCHEMBL4294688 0.87 PDE10A (0.43) PDE10AFPR1FPR2USP30AAK1
SCHEMBL4294928 0.84 ALDH1A1 (0.50) PDE10AMAPT
SCHEMBL6207573 0.83 FPR1 (0.41) PDE10AFPR1FPR2USP30AAK1
SCHEMBL12530374 0.83 HSD17B1 (0.47) PDE10AFPR1FPR2USP30AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240299348-A1 MODULATORS OF TRPML, THEIR COMPOSITIONS AND METHODS OF USE CARAWAY THERAPEUTICS, INC. 2024-09-12 US disclosed
WO-2022150461-A1 MODULATORS OF TRPML, THEIR COMPOSITIONS AND METHODS OF USE CARAWAY THERAPEUTICS, INC. (US) 2022-07-14 WO disclosed
WO-2022150461-A1 MODULATORS OF TRPML, THEIR COMPOSITIONS AND METHODS OF USE CARAWAY THERAPEUTICS, INC. (US) 2022-07-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240299348-A1 MODULATORS OF TRPML, THEIR COMPOSITIONS AND METHODS OF USE TRPM5, TRPM6, TRPM2 PDE10A 980/4885FPR1 3830/4885FPR2 3681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.