SCHEMBL28508679

SCHEMBL28508679

CN1CCN(c2ccc(-c3cnc4[nH]ccc4n3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 8/20 0.59
RIPK1 Q13546 1/20 0.57
RPS6KA3 P51812 7/20 0.53
MAP4K1 Q92918 1/20 0.53
KDM4E B2RXH2 1/20 0.52
NPC1 O15118 1/20 0.52
MAPT P10636 1/20 0.52
XBP1 P17861 1/20 0.52
RAB9A P51151 1/20 0.52
KLF5 Q13887 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
DYRK1A Q13627 1/20 0.52
CHEK1 O14757 2/20 0.49
RPS6KB1 P23443 1/20 0.48
FLT3 P36888 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28502461 0.89 MAPK1 (0.50) MAPK1RIPK1RPS6KA3MAP4K1KDM4E
SCHEMBL28503440 0.84 MAPK1 (0.54) MAPK1RIPK1RPS6KA3MAP4K1DYRK1A
SCHEMBL28513749 0.83 MAPK1 (0.54) MAPK1RIPK1MAP4K1NPC1DYRK1A
SCHEMBL30641871 0.83 MAPK1 (0.54) MAPK1RIPK1MAP4K1NPC1DYRK1A
SCHEMBL28510087 0.81 MAP3K11 (0.55) MAPK1RIPK1FLT3
SCHEMBL28504401 0.81 MAPK1 (0.55) MAPK1RIPK1DYRK1A
SCHEMBL28513878 0.81 MAPK1 (0.50) MAPK1RIPK1
SCHEMBL28905280 0.79 MAPK1 (0.53) MAPK1RIPK1MAPTRAB9ADYRK1A
SCHEMBL28514963 0.79 MAPK1 (0.53) MAPK1RIPK1MAPTRAB9ADYRK1A
SCHEMBL28499630 0.78 FLT3 (0.56) RIPK1RPS6KA3MAP4K1DYRK1ACHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed