SCHEMBL28513749

SCHEMBL28513749

Cc1cc(-c2cnc3[nH]ccc3n2)ccc1N1CCN(C)CC1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 13/20 0.54
DYRK1A Q13627 2/20 0.51
RIPK1 Q13546 1/20 0.49
PIK3CD O00329 1/20 0.47
PIK3R1 P27986 1/20 0.47
PIK3CA P42336 1/20 0.47
PIK3CG P48736 1/20 0.47
MAP4K1 Q92918 1/20 0.42
JAK2 O60674 2/20 0.42
JAK3 P52333 2/20 0.42
JAK1 P23458 1/20 0.42
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30641871 1.00 MAPK1 (0.54) MAPK1DYRK1ARIPK1PIK3CDPIK3R1
SCHEMBL28504401 0.87 MAPK1 (0.55) MAPK1DYRK1ARIPK1PIK3CDPIK3R1
SCHEMBL28513876 0.85 MAPK1 (0.55) MAPK1DYRK1ARIPK1MAP4K1
SCHEMBL28514903 0.85 MAPK1 (0.51) MAPK1DYRK1ARIPK1JAK2JAK3
SCHEMBL28508679 0.83 MAPK1 (0.59) MAPK1DYRK1ARIPK1MAP4K1NPC1
SCHEMBL28506118 0.82 DYRK1A (0.51) MAPK1DYRK1ARIPK1PIK3CDPIK3CA
SCHEMBL28507472 0.79 MAP4K1 (0.49) MAPK1MAP4K1JAK2JAK3
SCHEMBL28507725 0.78 RPS6KA3 (0.52) MAPK1MAP4K1JAK1
SCHEMBL28513565 0.77 MAPK1 (0.53) MAPK1DYRK1ARIPK1PIK3CDPIK3R1
SCHEMBL22858967 0.76 PIK3CD (0.52) MAPK1DYRK1ARIPK1PIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed