SCHEMBL28508682

SCHEMBL28508682

COc1ccc(C2=CCN(C)CC2)c(C#N)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.57
DRD2 P14416 2/20 0.47
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 1/20 0.45
QDPR P09417 1/20 0.44
DRD1 P21728 1/20 0.42
DRD5 P21918 1/20 0.42
DRD3 P35462 1/20 0.42
NOS2 P35228 1/20 0.42
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
RUNX1 Q01196 1/20 0.41
CBFB Q13951 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5536929 0.82 SLC6A4 (0.61) SLC6A4DRD2KMT2AALDH1A1QDPR
SCHEMBL28517116 0.81 SLC6A4 (0.55) SLC6A4DRD2DRD1
SCHEMBL23551386 0.81 SLC6A4 (0.49) SLC6A4QDPRALOX15
SCHEMBL30863499 0.79 SLC6A4 (0.43) SLC6A4QDPR
SCHEMBL27195917 0.79 SLC6A4 (0.43) SLC6A4QDPR
Hydrochloric Acid SCHEMBL31556090 0.76 QDPR (0.62) SLC6A4KMT2AALDH1A1QDPR
SCHEMBL5546728 0.75 QDPR (0.64) SLC6A4KMT2AALDH1A1QDPR
SCHEMBL31733726 0.74 SLC6A4 (0.55) SLC6A4DRD2KMT2AALDH1A1QDPR
SCHEMBL31733367 0.74 SLC6A4 (0.55) SLC6A4DRD2KMT2AALDH1A1QDPR
SCHEMBL7704740 0.73 SLC6A4 (1.00) SLC6A4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed