SCHEMBL2851001

SCHEMBL2851001

COc1ccc(CCc2ccc(CN(C(=O)CCC3CCCC3)c3ccc4c(c3)OC(C)(C)OC4=O)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 2/20 0.39
TRPM8 Q7Z2W7 1/20 0.37
OPRM1 P35372 2/20 0.37
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
SIRT5 Q9NXA8 1/20 0.36
STAT3 P40763 1/20 0.36
NR1H4 Q96RI1 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
RNF4 P78317 1/20 0.36
CHRM1 P11229 2/20 0.35
CHRM3 P20309 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853674 0.93 LTB4R2 (0.37) LTB4R2ALDH1A1KMT2AMEN1LMNA
SCHEMBL2850998 0.92 LTB4R2 (0.37) LTB4R2ALDH1A1KMT2AMEN1LMNA
SCHEMBL2861742 0.92 SLC6A4 (0.37) LTB4R2ALDH1A1PTGDR2SLC6A4
SCHEMBL2861774 0.91 GAA (0.38) LTB4R2KMT2AMEN1LMNASLC6A4
SCHEMBL13711758 0.88 SLC6A4 (0.41) LTB4R2ALDH1A1SLC6A4
SCHEMBL2851580 0.87 STAT3 (0.36) OPRM1ALDH1A1KMT2AMEN1MAPK1
SCHEMBL4457062 0.86 SLC6A4 (0.35) LTB4R2ALDH1A1PTGDR2SLC6A4
SCHEMBL13711662 0.86 SLC6A4 (0.41) LTB4R2SLC6A4
SCHEMBL13711754 0.86 LTB4R2 (0.43) LTB4R2SLC6A4
SCHEMBL2861740 0.85 SLC6A4 (0.34) LTB4R2OPRM1ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654247-B1 ALKYNYL ARYL CARBOXAMIDES MERCK SERONO SA (CH) 2010-01-20 EP disclosed