SCHEMBL28510034

SCHEMBL28510034

COc1cc(C=NNC(=O)c2ccc([N+](=O)[O-])cc2)ccc1O

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 9/20 0.79
MAPT P10636 7/20 0.79
POLB P06746 3/20 0.79
KDM4E B2RXH2 3/20 0.71
CA12 O43570 1/20 0.71
CA1 P00915 1/20 0.71
CA2 P00918 1/20 0.71
CA9 Q16790 1/20 0.71
MPO P05164 1/20 0.69
NT5E P21589 1/20 0.69
CYP3A4 P08684 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2C19 P33261 1/20 0.68
L3MBTL1 Q9Y468 1/20 0.68
ALDH1A1 P00352 2/20 0.67
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
LMNA P02545 1/20 0.67
TDP1 Q9NUW8 1/20 0.67
IKBKB O14920 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28515982 0.91 MAPT (0.79) GAAMAPTPOLBKDM4EMPO
SCHEMBL28513870 0.91 GAA (0.82) GAAMAPTPOLBKDM4ECA12
SCHEMBL28517560 0.88 MAPT (1.00) GAAMAPTPOLBKDM4ECYP3A4
SCHEMBL28516030 0.87 GAA (0.73) GAAMAPTPOLBKDM4ECA12
SCHEMBL3970958 0.86 MAPT (0.68) GAAMAPTPOLBKDM4ECYP3A4
SCHEMBL14417610 0.86 MAPT (0.68) GAAMAPTPOLBKDM4ECYP3A4
SCHEMBL3970964 0.86 MAPT (0.68) GAAMAPTPOLBKDM4ECYP3A4
SCHEMBL28515502 0.86 GAA (0.81) GAAMAPTPOLBKDM4ECA12
SCHEMBL28515978 0.86 GAA (0.81) GAAMAPTPOLBKDM4ECA12
SCHEMBL28506872 0.85 GAA (0.70) GAAMAPTPOLBKDM4ECA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN claimed
CN-112079744-B Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2021-07-30 CN disclosed
CN-112079744-A Aromatic acylhydrazone derivatives and application thereof as NA (adenosine) inhibitor 湖南大学 2020-12-15 CN disclosed