SCHEMBL28511552

SCHEMBL28511552

CN(C(=O)c1ccc(B2OC(C)(C)C(C)(C)O2)cc1)C1CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HB P07237 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CA1 P00915 6/20 0.41
CA2 P00918 6/20 0.41
CA9 Q16790 6/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALOX5 P09917 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
LPL P06858 3/20 0.41
LIPG Q9Y5X9 3/20 0.41
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALOX15 P16050 1/20 0.40
PDK2 Q15119 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499992 0.94 HSD11B1 (0.43) P4HBNPC1RAB9ACA1CA2
SCHEMBL28906215 0.94 HSD11B1 (0.43) P4HBNPC1RAB9ACA1CA2
SCHEMBL28499994 0.94 HSD11B1 (0.43) P4HBNPC1RAB9ACA1CA2
SCHEMBL16625305 0.90 MCHR1 (0.43) ALDH1A1PDK2
SCHEMBL16625313 0.87 HRH3 (0.47) NPC1RAB9AALDH1A1ALOX15PDK2
SCHEMBL16625306 0.87 MCHR1 (0.42) P4HBCA1CA2CA9LPL
SCHEMBL16625307 0.85 MCHR1 (0.52)
SCHEMBL16625315 0.83 MCHR1 (0.45) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL16625316 0.82 USP30 (0.57)
SCHEMBL1290961 0.82 P4HB (0.48) P4HBCA1CA2CA9LPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed