SCHEMBL28512074

SCHEMBL28512074

C[C@]1(O)CC[C@H](NC(=O)c2ccc(Br)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.50
NPC1 O15118 5/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
HPGD P15428 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C19 P33261 1/20 0.49
HPGDS O60760 1/20 0.48
MMP2 P08253 1/20 0.48
KMT2A Q03164 3/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 2/20 0.44
ALOX12 P18054 1/20 0.44
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28512075 1.00 RAB9A (0.50) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL28513976 1.00 RAB9A (0.50) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL3135552 0.84 RAB9A (0.62) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL17185341 0.80 NPC1 (0.62) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4770266 0.80 NPC1 (0.67) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL4768172 0.79 NPC1 (0.70) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL2254501 0.79 NPC1 (0.70) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL11920884 0.77 DEGS1 (0.46) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL28503436 0.77 MMP2 (0.42) RAB9ANPC1SMN1; SMN2HPGDCYP1A2
SCHEMBL28503437 0.77 MMP2 (0.42) RAB9ANPC1SMN1; SMN2HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed