SCHEMBL28512145

SCHEMBL28512145

COc1cc(Cl)ccc1C1=CCN(C)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.55
QDPR P09417 1/20 0.52
HTR6 P50406 1/20 0.48
DRD2 P14416 4/20 0.47
DRD4 P21917 1/20 0.47
TGFBR1 P36897 1/20 0.46
ACVR1 Q04771 1/20 0.46
CHRM1 P11229 2/20 0.45
DRD1 P21728 2/20 0.45
CHRM3 P20309 1/20 0.45
EHMT2 Q96KQ7 1/20 0.43
EHMT1 Q9H9B1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5536929 0.84 SLC6A4 (0.61) SLC6A4QDPRDRD2TGFBR1ACVR1
SCHEMBL27977286 0.80 QDPR (0.55) SLC6A4QDPRTGFBR1ACVR1EHMT2
SCHEMBL5547709 0.79 QDPR (0.54) SLC6A4QDPRHTR6DRD2DRD4
SCHEMBL28510095 0.78 SLC6A4 (0.60) SLC6A4QDPRDRD2TGFBR1ACVR1
SCHEMBL28517116 0.77 SLC6A4 (0.55) SLC6A4HTR6DRD2DRD4CHRM1
SCHEMBL10917066 0.77 SLC6A4 (0.58) SLC6A4QDPRHTR6DRD2DRD4
SCHEMBL4825697 0.76 CNR1 (0.54) QDPRHTR6
SCHEMBL31223021 0.75 QDPR (0.44) SLC6A4QDPRDRD2TGFBR1ACVR1
SCHEMBL7033282 0.74 QDPR (0.56) SLC6A4QDPRTGFBR1ACVR1EHMT2
Hydrochloric Acid SCHEMBL7030177 0.74 QDPR (0.56) SLC6A4QDPRTGFBR1ACVR1EHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed