SCHEMBL28512593

SCHEMBL28512593

c1ccc2c(c1)-c1ccncc1-2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.65
MAOB P27338 2/20 0.65
CYP19A1 P11511 2/20 0.45
CYP11B2 P19099 2/20 0.45
LIMK1 P53667 4/20 0.44
RPS6KA3 P51812 2/20 0.44
CDC25B P30305 1/20 0.44
TNF P01375 1/20 0.43
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2A6 P11509 2/20 0.39
NOTUM Q6P988 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
ACHE P22303 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19764657 1.00 MAOA (0.65) MAOAMAOBCYP19A1CYP11B2LIMK1
SCHEMBL14380259 1.00 MAOA (0.65) MAOAMAOBCYP19A1CYP11B2LIMK1
SCHEMBL12854062 0.88 RPS6KA3 (0.56) MAOAMAOBRPS6KA3TNFALDH1A1
SCHEMBL3066734 0.88 MAOA (0.87) MAOAMAOBLIMK1CDC25BALDH1A1
SCHEMBL12854064 0.88 RPS6KA3 (0.56) MAOAMAOBRPS6KA3TNFALDH1A1
SCHEMBL11369963 0.84 MAOA (0.50) MAOAMAOBCYP19A1CYP11B2TNF
SCHEMBL19013209 0.83 MAOA (0.87) MAOAMAOBCDC25BALDH1A1CYP3A4
SCHEMBL6926901 0.83 MAOA (0.95) MAOAMAOBCDC25BALDH1A1CYP1A2
SCHEMBL21726032 0.82 MAOA (0.48) MAOAMAOBCYP19A1CYP11B2LIMK1
SCHEMBL12854083 0.82 KDM4E (0.50) MAOAMAOBLIMK1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111777557-B Novel anti-tumor lead compound with aromatic biphenyl alkene as framework and application thereof 中国科学院上海有机化学研究所 2022-11-22 CN disclosed
CN-111777557-A Novel anti-tumor lead compound with aromatic biphenyl alkene as skeleton and application thereof 中国科学院上海有机化学研究所 2020-10-16 CN disclosed