SCHEMBL28514780

SCHEMBL28514780

COC(=O)c1ccc(-c2cncc(Br)c2)c(Cl)c1.O=C(O)c1ccc(-c2cncc(Br)c2)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH5 P11766 2/20 0.45
P4HTM Q9NXG6 1/20 0.43
POLB P06746 1/20 0.42
HCAR2 Q8TDS4 1/20 0.42
KDM4E B2RXH2 2/20 0.42
KDM6B O15054 1/20 0.42
KDM5C P41229 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM2A Q9Y2K7 1/20 0.42
KDM3A Q9Y4C1 1/20 0.42
CYP2A6 P11509 1/20 0.40
SRD5A2 P31213 1/20 0.40
MAPK1 P28482 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
SLC2A1 P11166 1/20 0.40
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21201422 0.95 CYP2A6 (0.43) KDM4ECYP2A6MAPK1MEN1ALDH1A1
SCHEMBL22977642 0.94 CYP2A6 (0.42) KDM4ECYP2A6MAPK1MEN1ALDH1A1
SCHEMBL21201466 0.90 ADH5 (0.52) ADH5P4HTMPOLBHCAR2SRD5A2
SCHEMBL6252933 0.79 SRD5A2 (0.59) ADH5KDM4EKDM6BKDM5CKDM4C
SCHEMBL23357794 0.77 PLAU (0.46) KDM4EMAPK1MEN1ALDH1A1MAPT
SCHEMBL22554086 0.76 CYP11B1 (0.51) KDM4EMAPK1MEN1ALDH1A1MAPT
SCHEMBL22977636 0.75 NOTUM (0.42) KDM4EMAPK1MEN1ALDH1A1MAPT
SCHEMBL3910111 0.75 EGFR (0.61) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL21201361 0.75 DHODH (0.48) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL21201316 0.74 ALPL (0.44) POLBKDM4EALDH1A1MAPTCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243374-A SREBP inhibitors comprising a 6-membered central ring 卡普勒斯疗法有限责任公司 2021-01-19 CN disclosed