SCHEMBL28516353

SCHEMBL28516353

COC(OC)c1nc(-c2ccc3c(cnn3C)c2)c(-c2cccc(C)n2)[nH]1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 19/20 0.60
MAPK14 Q16539 7/20 0.60
CYP1A2 P05177 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30183010 0.82 TGFBR1 (0.65) TGFBR1MAPK14CYP1A2
SCHEMBL4487787 0.82 TGFBR1 (0.47) TGFBR1MAPK14
SCHEMBL28510134 0.81 TGFBR1 (0.63) TGFBR1MAPK14CYP1A2
SCHEMBL28510984 0.80 TGFBR1 (0.59) TGFBR1MAPK14CYP1A2
SCHEMBL38661638 0.77 TGFBR1 (0.46) TGFBR1MAPK14
SCHEMBL22228617 0.77 TGFBR1 (0.40) TGFBR1MAPK14CYP1A2
SCHEMBL13680555 0.76 TGFBR1 (0.55) TGFBR1MAPK14
SCHEMBL6764903 0.76 TGFBR1 (0.66) TGFBR1MAPK14
SCHEMBL30182848 0.76 TGFBR1 (0.63) TGFBR1MAPK14CYP1A2
SCHEMBL22228605 0.75 TGFBR1 (0.47) TGFBR1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112266378-A Imidazole derivative containing indazole structure and preparation method and application thereof 延边大学 2021-01-26 CN claimed
CN-112266378-B Imidazole derivative containing indazole structure and preparation method and application thereof 延边大学 2021-10-12 CN disclosed
CN-112266378-A Imidazole derivative containing indazole structure and preparation method and application thereof 延边大学 2021-01-26 CN disclosed