SCHEMBL28516462

SCHEMBL28516462

O=C(NCC(c1ccccc1)n1cncn1)c1ccc2ccccc2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
KDM4C Q9H3R0 1/20 0.51
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
NPC1 O15118 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28497481 0.81 CYP24A1 (0.47) RAB9ASMN1; SMN2NPC1OPRM1DRD3
SCHEMBL28500074 0.80 CYP24A1 (0.62) GAAKDM4C
SCHEMBL28508999 0.77 CYP24A1 (0.68) ALDH1A1HPGDRAB9ASMN1; SMN2NFKB1
SCHEMBL22819409 0.72 GAA (0.66) GAAKDM4CALDH1A1MAPTHPGD
SCHEMBL28502275 0.71 RAB9A (0.52) ALDH1A1MAPTHPGDRAB9ASMN1; SMN2
SCHEMBL1220183 0.69 KDM4C (1.00) GAAKDM4CALDH1A1MAPTHPGD
SCHEMBL22819412 0.67 KDM4C (0.69) GAAKDM4CALDH1A1MAPTHPGD
SCHEMBL1742676 0.67 KDM4C (0.69) GAAKDM4CALDH1A1MAPTHPGD
SCHEMBL5095301 0.67 ALDH1A1 (0.73) GAAKDM4CALDH1A1MAPTHPGD
SCHEMBL6325976 0.67 CYP1A2 (0.52) GAAALDH1A1MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112194629-A Phenethyl azole derivative and preparation method and application thereof 聊城大学 2021-01-08 CN claimed
CN-112194629-B Phenethyl azole derivative and preparation method and application thereof 聊城大学 2023-10-24 CN disclosed
CN-112194629-A Phenethyl azole derivative and preparation method and application thereof 聊城大学 2021-01-08 CN disclosed