SCHEMBL28519302

SCHEMBL28519302

COC(=O)N1CC[C@@H](NC(=O)OCc2ccccc2)C1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.70
CTSL P07711 1/20 0.64
CTSB P07858 1/20 0.64
CTSK P43235 1/20 0.64
ALDH1A1 P00352 1/20 0.56
GAA P10253 1/20 0.56
DPP4 P27487 5/20 0.54
DPP7 Q9UHL4 5/20 0.54
KCNH2 Q12809 3/20 0.54
TSHR P16473 1/20 0.54
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
EPHX1 P07099 1/20 0.51
F13A1 P00488 2/20 0.50
TGM2 P21980 2/20 0.50
TGM1 P22735 2/20 0.50
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28519304 1.00 HSD11B1 (0.70) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL13161203 0.93 HSD11B1 (0.72) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL13243427 0.92 HSD11B1 (0.69) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL1191110 0.90 HSD11B1 (0.64) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL13740409 0.89 CTSL (0.68) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL3003867 0.89 CTSL (0.68) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL3667335 0.89 CTSL (0.68) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL6944572 0.89 HSD11B1 (0.65) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL951887 0.89 HSD11B1 (0.65) HSD11B1CTSLCTSBCTSKALDH1A1
SCHEMBL3726979 0.89 HSD11B1 (0.65) HSD11B1CTSLCTSBCTSKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188027-B Aromatic heterocyclic derivative and application thereof in medicine 广东东阳光药业有限公司 2020-10-20 CN disclosed