SCHEMBL28520243

SCHEMBL28520243

COC(=O)N1CCC(O)(CN)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.49
CYP2C9 P11712 3/20 0.46
USP2 O75604 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 7/20 0.43
CYP2C19 P33261 5/20 0.43
MAPK1 P28482 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 2/20 0.42
TSHR P16473 3/20 0.41
HIF1A Q16665 1/20 0.41
ALDH1A1 P00352 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL505705 0.84 L3MBTL1 (0.51) KMT2ATSHRALDH1A1
SCHEMBL154164 0.81 USP2 (0.49) USP2TSHR
SCHEMBL9181576 0.80 CYP2C9 (0.47) CYP2D6CYP2C9USP2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL17714540 0.80 USP2 (0.47) USP2TSHR
SCHEMBL1972942 0.76 SLC6A2 (0.33) CYP2D6USP2CYP1A2TSHRALDH1A1
SCHEMBL28515961 0.76 CYP2D6 (0.44) CYP2D6CYP2C9USP2CYP1A2CYP3A4
SCHEMBL22319499 0.76 HPGD (0.44) USP2MEN1KMT2AALDH1A1
SCHEMBL15451913 0.74 CYP1A2 (0.53) CYP2D6CYP2C9USP2CYP1A2CYP3A4
SCHEMBL3632294 0.72 CYP1A2 (0.56) CYP2D6CYP2C9USP2CYP1A2CYP3A4
SCHEMBL20617537 0.72 L3MBTL1 (0.53) CYP2D6CYP2C9USP2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188027-B Aromatic heterocyclic derivative and application thereof in medicine 广东东阳光药业有限公司 2020-10-20 CN disclosed