SCHEMBL28522018

SCHEMBL28522018

COc1cc2ncnc(Nc3cc(OCc4ccccc4)c(OC)cc3/C=C/C(=O)O)c2cc1O

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.56
RET P07949 9/20 0.52
KIF5B P33176 6/20 0.50
ERBB2 P04626 1/20 0.50
ERBB4 Q15303 1/20 0.50
KDR P35968 6/20 0.48
AURKB Q96GD4 2/20 0.48
AURKA O14965 1/20 0.47
PTGER4 P35408 1/20 0.47
PTGER2 P43116 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28522615 0.90 EGFR (0.57) EGFRRETKIF5BERBB2ERBB4
SCHEMBL28530529 0.87 EGFR (0.54) EGFRRETKIF5BKDR
SCHEMBL28518401 0.86 EGFR (0.53) EGFRERBB2KDR
SCHEMBL28529605 0.86 EGFR (0.53) EGFRERBB2ERBB4KDR
SCHEMBL28521215 0.85 EGFR (0.54) EGFRRETKIF5BERBB2ERBB4
SCHEMBL28908571 0.85 EGFR (0.53) EGFRRETKIF5BERBB2ERBB4
SCHEMBL28518408 0.84 EGFR (0.51) EGFRERBB2ERBB4KDR
SCHEMBL28521195 0.84 KDR (0.65) EGFRRETKIF5BKDRAURKB
SCHEMBL28527871 0.84 EGFR (0.51) EGFRERBB2ERBB4KDR
SCHEMBL28529600 0.83 PTGER4 (0.49) EGFRPTGER4PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808031-B Ferulic acid derivative and preparation method and application thereof 湖南中医药大学 2022-01-14 CN disclosed
CN-111808031-A Ferulic acid derivative and preparation method and application thereof 湖南中医药大学 2020-10-23 CN disclosed