SCHEMBL28908571

SCHEMBL28908571

COc1cc2ncnc(Nc3cc(/C=C/C(=O)O)cc(OC)c3OCc3ccccc3)c2cc1O

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.53
ERBB4 Q15303 2/20 0.49
ERBB2 P04626 1/20 0.49
RET P07949 5/20 0.48
AURKB Q96GD4 2/20 0.47
KIF5B P33176 2/20 0.46
AURKA O14965 1/20 0.46
APP P05067 1/20 0.46
ABCG2 Q9UNQ0 2/20 0.45
KDR P35968 1/20 0.45
ABCB1 P08183 1/20 0.45
RAF1 P04049 2/20 0.45
BRAF P15056 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28535568 0.86 EGFR (0.51) EGFRRETKIF5BKDR
SCHEMBL28522716 0.85 KDR (0.50) EGFRERBB2KDR
SCHEMBL28908582 0.85 EGFR (0.50) EGFRERBB4ERBB2KDR
SCHEMBL28522018 0.85 EGFR (0.56) EGFRERBB4ERBB2RETAURKB
SCHEMBL28516630 0.84 EGFR (0.49) EGFRERBB2KDR
SCHEMBL28522398 0.84 EGFR (0.49) EGFRERBB2KDR
SCHEMBL28524165 0.84 KDR (0.62) EGFRRETAURKBKIF5BAURKA
SCHEMBL28521215 0.82 EGFR (0.54) EGFRERBB4ERBB2RETAURKB
SCHEMBL6165317 0.79 EGFR (0.73) EGFRERBB4ERBB2RETAURKB
SCHEMBL6165325 0.79 EGFR (0.73) EGFRERBB4ERBB2RETAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808031-B Ferulic acid derivative and preparation method and application thereof 湖南中医药大学 2022-01-14 CN disclosed
CN-111808031-A Ferulic acid derivative and preparation method and application thereof 湖南中医药大学 2020-10-23 CN disclosed