SCHEMBL28522927

SCHEMBL28522927

NC(=O)C1(C(=O)N(c2ccccc2)c2ccc(O)c(F)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.52
ESR2 Q92731 3/20 0.52
ACHE P22303 1/20 0.36
PTGIR P43119 5/20 0.35
PTGDR Q13258 2/20 0.35
OPRK1 P41145 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
GRIN2B Q13224 3/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ADRA1A P35348 1/20 0.32
MCHR1 Q99705 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2152374 0.91 ESR1 (0.51) ESR1ESR2GRIN2BKDM4ELMNA
SCHEMBL19987724 0.90 ESR1 (0.43) ESR1ESR2PTGIRPTGDRKDM4E
SCHEMBL28515028 0.89 ESR1 (0.43) ESR1ESR2PTGIRPTGDR
SCHEMBL28517970 0.88 ESR1 (0.40) ESR1ESR2PTGIRPTGDRALDH1A1
SCHEMBL28515812 0.88 ESR1 (0.41) ESR1ESR2ACHEOPRK1GRIN2B
SCHEMBL558091 0.84 AGTR2 (0.41) ESR1ESR2PTGIRPTGDROPRK1
SCHEMBL28194894 0.83 NPSR1 (0.47) OPRK1NPSR1HSD17B10ALDH1A1
SCHEMBL2158816 0.81 ESR1 (0.41) ESR1ESR2KDM4ELMNAHSD17B10
SCHEMBL28514755 0.81 ACHE (0.46) ESR1ESR2ACHEGRIN2B
SCHEMBL28521626 0.79 ACHE (0.39) ESR1ESR2ACHEGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108503650-B Dioxane and quinazoline compound or medicinal salt or hydrate thereof and application of dioxane and quinazoline compound or medicinal salt or hydrate thereof as tyrosine kinase inhibitor 北京赛特明强医药科技有限公司 2021-02-12 CN disclosed