SCHEMBL28522962

SCHEMBL28522962

Clc1cccc(-c2nc(-c3ccccc3)cs2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.66
KDM4E B2RXH2 5/20 0.60
KMT2A Q03164 2/20 0.60
AR P10275 1/20 0.60
SREBF2 Q12772 2/20 0.57
HSD17B1 P14061 1/20 0.57
HSD17B2 P37059 1/20 0.57
MAPT P10636 2/20 0.56
RAB9A P51151 4/20 0.55
ALDH1A1 P00352 2/20 0.55
EIF4E P06730 1/20 0.55
CYP1A1 P04798 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP1B1 Q16678 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.53
LMNA P02545 2/20 0.53
MEN1 O00255 1/20 0.53
POLB P06746 1/20 0.53
GAA P10253 1/20 0.53
PKM P14618 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19196715 0.90 CYP19A1 (0.67) CYP19A1KDM4EKMT2AARSREBF2
SCHEMBL26121417 0.88 HSD17B1 (0.63) CYP19A1KDM4EKMT2ASREBF2HSD17B1
SCHEMBL12171802 0.84 CYP19A1 (0.67) CYP19A1KDM4EKMT2AHSD17B1HSD17B2
SCHEMBL4281217 0.83 RAB9A (0.75) CYP19A1KDM4EKMT2AARSREBF2
SCHEMBL11455457 0.83 RAB9A (0.75) CYP19A1KDM4EKMT2AARSREBF2
SCHEMBL31678026 0.82 MAPT (0.72) CYP19A1KDM4EKMT2AHSD17B1HSD17B2
SCHEMBL26136626 0.82 MAPT (0.72) CYP19A1KDM4EKMT2AHSD17B1HSD17B2
SCHEMBL31677707 0.82 MAPT (0.72) CYP19A1KDM4EKMT2AHSD17B1HSD17B2
SCHEMBL26135516 0.82 MAPT (0.72) CYP19A1KDM4EKMT2AHSD17B1HSD17B2
SCHEMBL2781370 0.82 KDM4E (0.85) CYP19A1KDM4EKMT2AARSREBF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110204507-B Process for producing 2-aryl-4-alkylthiazole compound 浙江大学 2021-03-02 CN disclosed