SCHEMBL2852406

SCHEMBL2852406

COc1cc(CCC(=O)CC(=O)O)cc(OC)c1O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 7/20 0.70
NFKB1 P19838 1/20 0.60
NFKB2 Q00653 1/20 0.60
RELA Q04206 1/20 0.60
OR51E2 Q9H255 1/20 0.59
LTA4H P09960 1/20 0.49
TNKS2 Q9H2K2 2/20 0.49
AKR1B1 P15121 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA3 P07451 1/20 0.47
PKM P14618 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
CA5A P35218 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
CA5B Q9Y2D0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL490990 0.86 ALOX5 (0.69) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL3756959 0.84 ALOX5 (0.71) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL4005549 0.83 ALOX5 (0.86) ALOX5NFKB1OR51E2LTA4HCYP1A2
SCHEMBL20940489 0.83 ALOX5 (1.00) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL10879308 0.83 ALOX5 (0.66) ALOX5OR51E2CA12CA1CA2
SCHEMBL13055954 0.82 ALOX5 (0.59) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL490925 0.81 ALOX5 (0.62) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL25363485 0.80 ALOX5 (0.60) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL29832717 0.80 ALOX5 (0.64) ALOX5NFKB1NFKB2RELAOR51E2
SCHEMBL24510591 0.79 ALOX5 (0.59) ALOX5NFKB1NFKB2RELAOR51E2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2195323-B1 Polyspirane compounds, use thereof in the treatment of malaria or toxoplasmosis and method for their preparation UNIV JOSEPH FOURIER (FR) 2011-12-28 EP disclosed
EP-2195323-A2 NOVEL POLYSPIRANE COMPOUNDS, APPLICATION THEREOF IN THE TREATMENT OF MALARIA OR TOXOPLASMOSIS AND METHOD FOR PREPARING SAME Université Joseph Fourier (FR) 2010-06-16 EP disclosed
WO-2009077677-A2 NOVEL POLYSPIRANE COMPOUNDS, APPLICATION THEREOF IN THE TREATMENT OF MALARIA OR TOXOPLASMOSIS AND METHOD FOR PREPARING SAME UNIVERSITE JOSEPH FOURIER (FR) 2009-06-25 WO disclosed