Arbutin

Arbutin

SCHEMBL285242

OC[C@H]1OC(Oc2ccc(O)cc2)[C@H](O)[C@@H](O)[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TYR

The experimentally established mechanism targets of Arbutin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TYR known ✓ P14679 4/20 1.00
POLB P06746 2/20 0.67
KDM4E B2RXH2 1/20 0.67
GAA P10253 1/20 0.67
MAPT P10636 1/20 0.67
G6PD P11413 1/20 0.67
MAPK1 P28482 1/20 0.67
ADRA1A P35348 1/20 0.67
PTGS2 P35354 1/20 0.67
NPC1 O15118 1/20 0.59
ALDH1A2 O94788 1/20 0.59
ALDH2 P05091 1/20 0.59
ALDH1B1 P30837 1/20 0.59
RAB9A P51151 1/20 0.59
IL2 P60568 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
AKR1B1 P15121 1/20 0.59
DPP4 P27487 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Arbutin SCHEMBL13313589 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL4289558 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL15481351 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL13956277 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL18175043 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL36352 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL5438300 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL12998301 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL13054606 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT
Arbutin SCHEMBL435261 1.00 TYR (1.00) TYRPOLBKDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 236 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114425024-A Stabilized compositions containing hydroquinone or derivatives thereof 株式会社LG生活健康 2022-05-03 CN claimed
CN-111393492-B Alkyne-alkene hydroquinone glucoside, preparation method thereof and application of alkyne-alkene hydroquinone glucoside in preparation of liver X receptor agonist 中国科学院南海海洋研究所 2021-06-11 CN claimed
CN-111870555-A Anti-aging repair essence and preparation process thereof 江苏奥普莱医疗用品有限公司 2020-11-03 CN claimed
CN-111393492-A Alkyne-alkene hydroquinone glucoside, preparation method thereof and application of alkyne-alkene hydroquinone glucoside in preparation of liver X receptor agonist 中国科学院南海海洋研究所 2020-07-10 CN claimed
CN-1849390-A High level production of arbutin in green plants and microbes DU PONT (US) 2006-10-18 CN claimed
US-7056742-B2 High Level production of arbutin in green plants E. I. DU PONT DE NEMOURS AND COMPANY (US) 2006-06-06 US claimed
WO-2004113504-A2 HIGH LEVEL PRODUCTION OF ARBUTIN IN GREEN PLANTS AND MICROBES E.I. DUPONT DE NEMOURS AND COMPANY (US) 2004-12-29 WO claimed
US-20040261147-A1 High level production of arbutin in green plants and microbes UNIVERSITY OF NORTH TEXAS 2004-12-23 US claimed
JP-9175987-A None JP disclosed
JP-61225106-A None JP disclosed
JP-7206632-A None JP disclosed
JP-61225112-A None JP disclosed
JP-6009366-A None JP disclosed
JP-9077654-A None JP disclosed
JP-H06107533-A COSMETIC POLA CHEM IND INC 1994-04-19 JP disclosed
JP-H069366-A EXTERNAL AGENT FOR SKIN SHISEIDO CO LTD 1994-01-18 JP disclosed
US-4764505-A GLYCOSIDE OF HYDROQUINONE-SUPPRESSION OF SKIN IRRITATION SHISEIDO COMPANY LTD. (JP) 1988-08-16 US disclosed
JP-S61225106-A DERMATIC AGENT FOR EXTERNAL USE SHISEIDO CO LTD 1986-10-06 JP disclosed
JP-S61225112-A HAIR COSMETIC SHISEIDO CO LTD 1986-10-06 JP disclosed
JP-S61225114-A DERMATIC AGENT FOR EXTERNAL USE SHISEIDO CO LTD 1986-10-06 JP disclosed