SCHEMBL28524201

SCHEMBL28524201

CC(C)(C)OC(=O)NC(Cc1c(F)cccc1Br)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 9/20 0.47
CTSK P43235 7/20 0.47
SCN9A Q15858 4/20 0.44
CTSB P07858 2/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
PTPN1 P18031 1/20 0.42
CYP3A4 P08684 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.42
CTSL P07711 1/20 0.41
AAK1 Q2M2I8 1/20 0.40
ACE P12821 1/20 0.40
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28523141 0.86 CTSS (0.47) CTSSCTSKCTSBALDH1A1MAPT
SCHEMBL28532406 0.86 CTSS (0.47) CTSSCTSKCTSBALDH1A1MAPT
SCHEMBL28523218 0.82 CTSS (0.44) CTSSCTSKCTSBALDH1A1MAPT
SCHEMBL4584520 0.81 PTPN1 (0.55) CTSSCTSKSCN9ACTSBPTPN1
SCHEMBL1529787 0.81 PTPN1 (0.55) CTSSCTSKSCN9ACTSBPTPN1
SCHEMBL30825600 0.81 CTSS (0.47) CTSSCTSKSCN9ACTSBPTPN1
SCHEMBL28989417 0.80 TACR1 (0.48) CTSSCTSKCTSBCTSLAAK1
SCHEMBL30681226 0.79 AAK1 (0.42) CTSSCTSKSCN9ACTSBALDH1A1
SCHEMBL30681530 0.79 AAK1 (0.42) CTSSCTSKSCN9ACTSBALDH1A1
SCHEMBL30825613 0.79 KLK5 (0.43) CTSSCTSKSCN9ACTSBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105916836-B Method for producing 2-fluoro-4-borono-L-phenylalanine and precursor thereof 斯特拉制药公司 2021-02-09 CN disclosed