SCHEMBL28524700

SCHEMBL28524700

COC(=O)c1ccnc2c1c(C=O)cn2Cc1ccc(OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90B1 P14625 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
CHRM1 P11229 3/20 0.39
AHR P35869 1/20 0.39
KDM4E B2RXH2 2/20 0.39
POLB P06746 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ASPH Q12797 1/20 0.39
KDM8 Q8N371 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1079929 0.81 CHRM1 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5052648 0.73 HSP90B1 (0.47) HSP90B1HDAC1HDAC6CHRM1AHR
SCHEMBL1953325 0.71 ATR (0.46) KDM4EPOLBALDH1A1GLAGAA
SCHEMBL1607759 0.70 HDAC6 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28525168 0.70 FGFR1 (0.40) KDM4EALDH1A1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL699995 0.70 APP (0.50) POLBL3MBTL1ALDH1A1SMN1; SMN2GAA
SCHEMBL21043082 0.70 L3MBTL1 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3802315 0.70 HSP90AA1 (0.51) HDAC4HDAC1HDAC2HDAC6CHRM1
SCHEMBL27988410 0.69 LMNA (0.40) KDM4EL3MBTL1ASPHKDM8ALDH1A1
SCHEMBL21518857 0.69 SMN1; SMN2 (0.45) HDAC1KDM4EL3MBTL1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112390799-B Nitrogen-containing heterocyclic 5-HT3 receptor regulator and preparation method and application thereof 科岭源生物科技(深圳)有限公司 2022-04-29 CN disclosed
CN-112390799-A Nitrogen-containing heterocyclic 5-HT3 receptor regulator and preparation method and application thereof 成都科岭源医药技术有限公司 2021-02-23 CN disclosed