SCHEMBL28524701

SCHEMBL28524701

O=[PH](OCc1ccc(C(F)(F)F)cc1F)OCc1ccc(C(F)(F)F)cc1F

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.61
DAO P14920 1/20 0.43
FFAR1 O14842 1/20 0.42
PDE2A O00408 2/20 0.37
AGXT P21549 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
BACE1 P56817 1/20 0.35
CES2 O00748 1/20 0.35
MPL P40238 1/20 0.35
SRD5A2 P31213 1/20 0.35
NAAA Q02083 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34
APP P05067 1/20 0.34
PTGER1 P34995 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28524703 0.87 IDO1 (0.58) IDO1DAOFFAR1PDE2AAGXT
SCHEMBL12516416 0.77 IDO1 (0.67) IDO1DAOFFAR1PDE2AAGXT
SCHEMBL16214946 0.77 IDO1 (0.67) IDO1DAOFFAR1PDE2AAGXT
SCHEMBL3156002 0.75 IDO1 (0.63) IDO1DAOFFAR1PDE2AAGXT
SCHEMBL6789942 0.74 IDO1 (0.58) IDO1DAOFFAR1PDE2ASLC6A4
SCHEMBL1117948 0.74 IDO1 (0.58) IDO1DAOFFAR1PDE2ASLC6A4
SCHEMBL7977134 0.74 IDO1 (0.62) IDO1DAOFFAR1PDE2ASLC6A4
SCHEMBL27634838 0.74 IDO1 (0.58) IDO1DAOFFAR1PDE2ASLC6A4
SCHEMBL19409499 0.74 IDO1 (0.58) IDO1DAOFFAR1PDE2ASLC6A4
SCHEMBL14255637 0.74 IDO1 (0.58) IDO1DAOFFAR1PDE2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114364684-A Heterocyclic compounds 豪夫迈·罗氏有限公司 2022-04-15 CN disclosed
CN-112867720-A Novel heterocyclic compounds as monoacylglycerol lipase inhibitors 豪夫迈·罗氏有限公司 2021-05-28 CN disclosed
CN-112469724-A Novel heterocyclic compounds as monoacylglycerol lipase inhibitors 豪夫迈·罗氏有限公司 2021-03-09 CN disclosed