SCHEMBL28526784

SCHEMBL28526784

Cc1nnc(-c2cccc(Oc3ccc(N(C(=O)O)C(C)(C)C)c(Cl)c3)c2)o1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.38
HPGD P15428 3/20 0.38
LMNA P02545 3/20 0.38
KMO O15229 1/20 0.38
KDM4E B2RXH2 3/20 0.38
TSHR P16473 3/20 0.37
GAA P10253 1/20 0.37
MAPK14 Q16539 3/20 0.37
MAPK11 Q15759 1/20 0.37
MAPT P10636 3/20 0.36
THRB P10828 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HTT P42858 2/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
CCR6 P51684 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CTSA P10619 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28538655 0.89 KDM4E (0.37) SMN1; SMN2HPGDLMNAKDM4ETSHR
SCHEMBL23355371 0.79 KDM4E (0.45) SMN1; SMN2HPGDLMNAKMOKDM4E
SCHEMBL21616262 0.77 KDM4E (0.41) SMN1; SMN2HPGDLMNAKDM4ETSHR
SCHEMBL30203153 0.77 KDM4E (0.41) SMN1; SMN2HPGDLMNAKDM4ETSHR
SCHEMBL28909804 0.74 KMO (0.47) SMN1; SMN2LMNAKMOKDM4EALDH1A1
SCHEMBL21612825 0.72 KDM4E (0.42) SMN1; SMN2HPGDLMNAKDM4ETSHR
SCHEMBL23355373 0.71 KDM4E (0.45) SMN1; SMN2HPGDLMNAKDM4ETSHR
SCHEMBL15117470 0.70 MAPK14 (0.37) HPGDLMNAKDM4ETSHRMAPK14
SCHEMBL1690753 0.69 ESR2 (0.45) MEN1KMT2A
SCHEMBL23368213 0.69 CYP17A1 (0.42) SMN1; SMN2KDM4EMAPTTHRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112334460-A Biaryl ether type quinazoline derivative 第一三共株式会社 2021-02-05 CN disclosed