SCHEMBL28526980

SCHEMBL28526980

O=C(O)c1cc2cc3c(cc2s1)CCCN3

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
MAPT P10636 1/20 0.50
GPR35 Q9HC97 3/20 0.49
ALDH1A1 P00352 2/20 0.47
DAO P14920 1/20 0.47
BCL2L1 Q07817 1/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
PTPN2 P17706 2/20 0.38
AR P10275 2/20 0.36
ATM Q13315 1/20 0.35
TBXAS1 P24557 3/20 0.34
GAA P10253 1/20 0.34
PLAU P00749 1/20 0.34
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830635 0.87 GPR35 (0.50) KDM4EMAPTGPR35ALDH1A1DAO
SCHEMBL19433653 0.86 PTPN2 (0.42) KDM4EMAPTGPR35ALDH1A1CA12
SCHEMBL19433627 0.78 CRBN (0.42) KDM4EMAPTALDH1A1PTPN2ATM
SCHEMBL28521802 0.78 GPR35 (0.47) KDM4EMAPTGPR35ALDH1A1DAO
SCHEMBL31672932 0.77 ATM (0.40) KDM4EMAPTALDH1A1CA12CA1
SCHEMBL4827429 0.73 PTPN2 (0.43) KDM4EMAPTGPR35ALDH1A1PTPN2
SCHEMBL28529829 0.73 RARB (0.46) GPR35ALDH1A1DAOBCL2L1PTPN2
SCHEMBL11359596 0.73 ALDH1A1 (0.54) KDM4EMAPTGPR35ALDH1A1DAO
SCHEMBL30643033 0.73 GPR35 (0.76) KDM4EMAPTGPR35ALDH1A1DAO
SCHEMBL20916098 0.69 CA12 (0.43) KDM4EMAPTALDH1A1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107001345-B Heterocyclic derivatives and use thereof 株式会社C&C新药研究所 2021-03-02 CN disclosed