SCHEMBL28527720

SCHEMBL28527720

OB(O)c1ccc(-c2cccc(F)c2)s1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 10/20 0.62
HSD17B2 P37059 10/20 0.62
ESRRG P62508 6/20 0.49
ESR2 Q92731 4/20 0.46
ESR1 P03372 3/20 0.46
CNR1 P21554 1/20 0.44
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
PRF1 P14222 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2556281 0.83 HSD17B1 (0.49) HSD17B1HSD17B2ESRRGESR2ESR1
SCHEMBL290143 0.83 HSD17B1 (0.48) HSD17B1HSD17B2CYP3A4CYP2C19
SCHEMBL28524259 0.81 MGLL (0.50) HSD17B1HSD17B2PRF1
SCHEMBL28529085 0.81 HSD17B1 (0.47) HSD17B1HSD17B2CNR1TP53MAPT
SCHEMBL12107122 0.79 HSD17B1 (0.50) HSD17B1HSD17B2ESR2ESR1CYP3A4
SCHEMBL20764241 0.79 HSD17B1 (0.72) HSD17B1HSD17B2ESRRGESR2CNR1
SCHEMBL28523476 0.77 HDAC6 (0.55) HSD17B1HSD17B2CNR1CYP3A4CYP2D6
SCHEMBL1179817 0.76 HSD17B1 (1.00) HSD17B1HSD17B2ESRRGESR2CYP3A4
SCHEMBL28519933 0.75 MGLL (0.47) HSD17B1HSD17B2ESR2ESR1PRF1
SCHEMBL14332594 0.74 HSD17B1 (0.61) HSD17B1HSD17B2ESRRGESR2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602834-B Bruton's tyrosine kinase inhibitor 北京盛诺基医药科技股份有限公司 2021-01-08 CN disclosed