SCHEMBL2852818

SCHEMBL2852818

Cc1cccc(NC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
MAPT P10636 2/20 0.50
NR1H4 Q96RI1 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CCR1 P32246 1/20 0.50
BRAF P15056 1/20 0.50
NPY5R Q15761 1/20 0.49
MALT1 Q9UDY8 6/20 0.49
KMT2A Q03164 1/20 0.48
TP53 P04637 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
SCN2A Q99250 1/20 0.47
SCN10A Q9Y5Y9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850032 0.91 NPC1 (0.56) NPC1RAB9AMAPTNR1H4KDM4E
SCHEMBL13513708 0.88 KDM4E (0.53) MAPTKDM4EALDH1A1BRAFMALT1
SCHEMBL2857034 0.87 KDM4E (0.62) NPC1RAB9AMAPTNR1H4KDM4E
SCHEMBL2850892 0.87 NR1H4 (0.53) NPC1RAB9AMAPTNR1H4KDM4E
SCHEMBL14539344 0.87 KDM4E (0.52) MAPTNR1H4KDM4EALDH1A1BRAF
SCHEMBL13513684 0.86 CCR1 (0.54) MAPTNR1H4KDM4EALDH1A1CCR1
SCHEMBL13513752 0.86 BRAF (0.49) NPC1RAB9AMAPTNR1H4KDM4E
SCHEMBL14539343 0.85 NR1H4 (0.47) MAPTNR1H4KDM4EALDH1A1CCR1
SCHEMBL2850859 0.85 KEAP1 (0.51) MAPTNR1H4KDM4EALDH1A1BRAF
SCHEMBL2852325 0.85 KEAP1 (0.51) MAPTNR1H4KDM4EALDH1A1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed