SCHEMBL28528902

SCHEMBL28528902

Cc1cc2c(cc1[N+](=O)[O-])c(=O)c(Br)cn2C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.38
HTT P42858 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.37
POLB P06746 2/20 0.35
ALDH1A1 P00352 5/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
RECQL P46063 1/20 0.34
GAA P10253 2/20 0.34
HSP90AA1 P07900 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
CCR6 P51684 1/20 0.34
NLRP1 Q9C000 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30686055 1.00 MAPT (0.38) MAPTHTTNPSR1LMNAKDM4E
SCHEMBL30686034 0.82 CYP1A2 (0.35) MAPTHTTNPSR1LMNAKDM4E
SCHEMBL28534508 0.82 CYP1A2 (0.35) MAPTHTTNPSR1LMNAKDM4E
SCHEMBL28519693 0.80 LMNA (0.46) MAPTHTTLMNAKDM4EPOLB
SCHEMBL30686011 0.80 LMNA (0.46) MAPTHTTLMNAKDM4EPOLB
SCHEMBL28517539 0.77 ATAD2 (0.47) MAPTHTTKDM4EALDH1A1CYP3A4
SCHEMBL28362553 0.75 MAPT (0.49) MAPTNPSR1LMNACYP1A2POLB
SCHEMBL28521783 0.75 POLB (0.62) MAPTNPSR1LMNAKDM4EPOLB
SCHEMBL17579519 0.70 LMNA (0.39) MAPTHTTNPSR1LMNAKDM4E
SCHEMBL2442735 0.69 CYP1A2 (0.53) MAPTCYP1A2ALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409332-B Triazole derivative and application thereof in medicines 广东东阳光药业股份有限公司 2023-12-08 CN disclosed
CN-112409332-A Triazole derivative and application thereof in medicines 广东东阳光药业有限公司 2021-02-26 CN disclosed