SCHEMBL28529

SCHEMBL28529

Sn1cnc2cncnc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.42
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
LTA4H P09960 1/20 0.36
CYP1A2 P05177 12/20 0.36
CYP3A4 P08684 9/20 0.36
ALDH1A1 P00352 8/20 0.36
CYP2C19 P33261 7/20 0.36
TSHR P16473 7/20 0.36
CYP2C9 P11712 7/20 0.36
LMNA P02545 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HBB P68871 1/20 0.36
MKNK2 Q9HBH9 1/20 0.35
USP2 O75604 6/20 0.34
CLK4 Q9HAZ1 4/20 0.33
CYP2D6 P10635 2/20 0.33
HSD17B10 Q99714 3/20 0.32
MAPK1 P28482 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL316719 0.98 FDPS (0.41) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL28659170 0.98 FDPS (0.41) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL671498 0.98 FDPS (0.41) FDPSHDAC1HDAC6LTA4HCYP1A2
Tetrahydrofuran SCHEMBL28855131 0.86 FDPS (0.35) FDPSHDAC1HDAC6LTA4HCYP1A2
Malonic Acid SCHEMBL28513650 0.85 HDAC1 (0.44) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL28340215 0.76 FDPS (0.44) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL28779724 0.74 FDPS (0.42) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL7787139 0.74 FDPS (0.42) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL30341176 0.74 GRM5 (0.46) FDPSHDAC1HDAC6LTA4HCYP1A2
SCHEMBL28763050 0.74 FDPS (0.46) FDPSHDAC1HDAC6LTA4HCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4033 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260138973-A1 SUBSTITUTED PYRIDINES FOR USE IN TREATING OR PREVENTING INFLAMMATORY DISEASES OR DISEASES ASSOCIATED WITH AN UNDESIRABLE IMMUNE RESPONSE SITRYX THERAPEUTICS LTD (GB) 2026-05-21 US claimed
US-20260137680-A1 NOVEL COMPOUNDS SITRYX THERAPEUTICS LTD (GB) 2026-05-21 US claimed
US-12617762-B2 Carboxy derivatives with antiinflamatory properties SITRYX THERAPEUTICS LIMITED (GB) 2026-05-05 US claimed
US-12618111-B2 Methods of diagnosing inflammatory bowel disease through RNASET2 CEDARS-SINAI MEDICAL CENTER (US) 2026-05-05 US claimed
US-20260085061-A1 PHTHALAZINE DERIVATIVES AS PYRUVATE KINASE MODULATORS SITRYX THERAPEUTICS LIMITED (GB) 2026-03-26 US claimed
EP-4714452-A1 METHODS FOR TREATING SARS COV-2 INFECTIONS Gilead Sciences, Inc. (US) 2026-03-25 EP claimed
EP-4081511-B3 CARBOXY DERIVATIVES WITH ANTIINFLAMMATORY PROPERTIES SITRYX THERAPEUTICS LTD (GB) 2026-03-04 EP claimed
US-12534571-B2 Amphiphilic block copolymer, preparation method thereof and nanomicelle drug-loading system SHANGHAI BEST-LINK BIOSCIENCE, LLC (CN) 2026-01-27 US claimed
US-20250367113-A1 DRUG DELIVERY SYSTEM COMPRISING AN ANTI-INFLAMMATORY AGENT OR A SALT THEREOF FOR THE APPLICATION TO ESOPHAGEAL MUCOUS MEMBRANES ESOCAP AG (CH) 2025-12-04 US claimed
EP-4634167-A1 SUBSTITUTED PYRIDINES FOR USE IN TREATING OR PREVENTING INFLAMMATORY DISEASES OR DISEASES ASSOCIATED WITH AN UNDESIRABLE IMMUNE RESPONSE Sitryx Therapeutics Limited (GB) 2025-10-22 EP claimed
WO-1997007201-A1 IDENTIFICATION OF TWO NOVEL MUTANT ALLELES OF HUMAN THIOPURINE S-METHYLTRANSFERASE, AND DIAGNOSTIC USES THEREOF ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 1997-02-27 WO claimed
EP-0754046-A1 USE OF PHOSPHONYLMETHOXYALKYL NUCLEOSIDES FOR THE TREATMENT OF RAISED INTRAOCULAR PRESSURE FREEMAN, William R. (US) 1997-01-22 EP claimed
WO-1996003653-A1 SUPERPARAMAGNETIC PARTICLES, PROCESS FOR THEIR PRODUCTION AND THEIR USE SILICA GEL GES.MBH ABSORPTIONSTECHNIK, APPARATEBAU (DE) 1996-02-08 WO claimed
US-5470737-A Isolation and purification of DNA sequence with code, genetic engineering MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 1995-11-28 US claimed
WO-1995026734-A1 USE OF PHOSPHONYLMETHOXYALKYL NUCLEOSIDES FOR THE TREATMENT OF RAISED INTRAOCULAR PRESSURE FREEMAN WILLIAM R (US) 1995-10-12 WO claimed
US-5120753-A Chemoprevention of electrophilic damage by mercaptopurine analogs BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1992-06-09 US claimed
EP-0478546-A1 CHEMOPREVENTION OF ELECTROPHILIC DAMAGE BY MERCAPTOPURINE ANALOGS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1992-04-08 EP claimed
WO-1990004966-A2 CHEMOPREVENTION OF ELECTROPHILIC DAMAGE BY MERCAPTOPURINE ANALOGS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1990-05-17 WO claimed
US-4075021-A COMPOUND WHICH RELEASES A SUBSTANCE WHICH PROMOTES BLEACHING OF DEVELOPED SILVER KONISHIROKU PHOTO INDUSTRY CO., LTD. (JA) 1978-02-21 US claimed
US-3939089-A PEROXYSULFATE TOKAI DENKA KOGYO KABUSHIKI KAISHA (JA) 1976-02-17 US claimed