SCHEMBL28530840

SCHEMBL28530840

Cn1c(-c2cc3ccccc3n2CC2CC2)nc2cc(C=O)ccc21

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PADI4 Q9UM07 18/20 0.58
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
PTGER4 P35408 1/20 0.43
BRD4 O60885 1/20 0.41
BAZ2A Q9UIF9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28529826 0.99 PADI4 (0.57) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL30325275 0.86 PADI4 (0.52) PADI4PTGER4
SCHEMBL25145104 0.86 PADI4 (0.52) PADI4PTGER4
Hydrochloric Acid SCHEMBL28524626 0.85 PADI4 (0.53) PADI4PTGER4
Hydrochloric Acid SCHEMBL30325573 0.85 PADI4 (0.53) PADI4PTGER4
SCHEMBL28539904 0.83 LMNA (0.47) PADI4BRD4
SCHEMBL28539969 0.82 PADI4 (0.61) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL18247356 0.82 PADI4 (0.69) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL28561906 0.82 PADI4 (0.45) PADI4
SCHEMBL28539017 0.82 KMT2A (0.44) PADI4PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849015-B Benzimidazole derivatives as PAD4 inhibitors 葛兰素知识产权发展有限公司 2021-03-19 CN claimed
CN-107849015-B Benzimidazole derivatives as PAD4 inhibitors 葛兰素知识产权发展有限公司 2021-03-19 CN disclosed