SCHEMBL2853112

SCHEMBL2853112

O=C(NCCN1CCOCC1)Nc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.58
CNR1 P21554 2/20 0.58
LMNA P02545 3/20 0.57
KMT2A Q03164 1/20 0.57
ALDH1A1 P00352 2/20 0.49
HTR1A P08908 1/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
KCNH2 Q12809 1/20 0.49
CD274 Q9NZQ7 1/20 0.49
ABCB1 P08183 1/20 0.49
EPHX2 P34913 4/20 0.48
KDM4E B2RXH2 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
ALOX15 P16050 1/20 0.47
HTT P42858 1/20 0.47
MAPK1 P28482 2/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850703 0.91 CNR1 (0.56) SMN1; SMN2CNR1LMNAKMT2AALDH1A1
SCHEMBL2859857 0.90 CNR1 (0.55) SMN1; SMN2CNR1LMNAKMT2AALDH1A1
SCHEMBL2880891 0.81 CNR1 (0.54) SMN1; SMN2CNR1LMNAKMT2AKDM4E
SCHEMBL2860983 0.80 MAPT (0.49) SMN1; SMN2LMNAKMT2AALDH1A1EPHX2
SCHEMBL2858063 0.80 MAPT (0.57) SMN1; SMN2LMNAALDH1A1KDM4EMAPT
SCHEMBL2862263 0.79 MAPT (0.47) CNR1LMNAALDH1A1KDM4EMAPT
SCHEMBL2856146 0.79 CNR1 (0.53) SMN1; SMN2CNR1LMNAKMT2AALDH1A1
SCHEMBL2872664 0.78 MALT1 (0.42) MAPT
SCHEMBL2854478 0.78 ITGB3 (0.46) SMN1; SMN2LMNAKMT2AMAPTGAA
SCHEMBL2856795 0.78 NPC1 (0.46) CNR1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed