SCHEMBL28533682

SCHEMBL28533682

O=C(O)c1ccc(N2CC(c3ccc(C(F)(F)F)cc3)C[C@@H]2COC(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.39
PTGER4 P35408 4/20 0.35
F2R P25116 4/20 0.35
LTA4H P09960 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
OPRD1 P41143 1/20 0.35
P2RY14 Q15391 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
NOTUM Q6P988 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCR2 P41597 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28540107 1.00 SRD5A2 (0.39) SRD5A2PTGER4F2RLTA4HPSEN1
SCHEMBL23631891 1.00 SRD5A2 (0.39) SRD5A2PTGER4F2RLTA4HPSEN1
SCHEMBL28537484 0.91 SRD5A2 (0.38) SRD5A2PTGER4LTA4HPSEN1PSEN2
SCHEMBL21616610 0.91 SRD5A2 (0.38) SRD5A2PTGER4F2RLTA4HPSEN1
SCHEMBL28529305 0.91 SRD5A2 (0.38) SRD5A2PTGER4LTA4HPSEN1PSEN2
SCHEMBL21619810 0.91 MAOB (0.38) F2RPSEN1PSEN2APH1BNCSTN
SCHEMBL28542902 0.89 KDM4E (0.42) F2RCCR2KCNH2
SCHEMBL23632260 0.89 KDM4E (0.42) F2RCCR2KCNH2
SCHEMBL28910602 0.88 FPR1 (0.41) SRD5A2PTGER4F2RLTA4HADRA2A
SCHEMBL28532591 0.87 SRD5A2 (0.36) SRD5A2PTGER4F2RLTA4HPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed