SCHEMBL28534201

SCHEMBL28534201

Nc1cccc2c3ccccc3c3ccc4ccccc4c3c12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 6/20 0.58
ALDH1A1 P00352 6/20 0.58
HPGD P15428 4/20 0.58
TSHR P16473 4/20 0.58
CYP3A4 P08684 3/20 0.58
KEAP1 Q14145 1/20 0.58
CYP1A2 P05177 2/20 0.54
THRB P10828 1/20 0.54
HPRT1 P00492 4/20 0.53
TDP1 Q9NUW8 2/20 0.44
CYP2A6 P11509 1/20 0.44
HIF1A Q16665 2/20 0.44
ERBB2 P04626 1/20 0.44
FYN P06241 1/20 0.44
MAOA P21397 1/20 0.44
ACHE P22303 1/20 0.44
AHR P35869 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18600581 0.90 HSD17B10 (0.58) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL16194308 0.88 ALDH1A1 (0.60) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL31158232 0.85 ALDH1A1 (0.65) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL3630203 0.85 ALDH1A1 (0.65) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL18600593 0.84 ALDH1A1 (0.52) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL1038972 0.84 HPRT1 (0.72) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL29697319 0.84 HPRT1 (0.72) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL29518611 0.83 ALDH1A1 (0.62) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL28712139 0.83 ALDH1A1 (0.62) HSD17B10ALDH1A1HPGDTSHRCYP3A4
SCHEMBL8968929 0.82 HPRT1 (0.68) HSD17B10ALDH1A1HPGDTSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110194741-B 4-benzoyl piperazine-3-nitro-1, 8-naphthalimide derivative and preparation method and application thereof 桂林医学院 2022-09-09 CN disclosed
CN-110194740-B 4-tert-butyloxycarbonylpiperazine-1, 8-naphthalimide derivative and synthetic method and application thereof 桂林医学院 2022-06-17 CN disclosed
CN-112472699-A Combination methods for improving the therapeutic benefit of bisantrene and derivatives 种族肿瘤学公司 2021-03-12 CN disclosed