SCHEMBL2853700

SCHEMBL2853700

Nc1cnc2ccccc2c1.Nc1ncccn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
HSP90AA1 P07900 2/20 0.56
MAPT P10636 2/20 0.56
ATM Q13315 2/20 0.56
KDM4E B2RXH2 1/20 0.56
TP53 P04637 1/20 0.56
HSP90AB1 P08238 1/20 0.56
TSHR P16473 1/20 0.56
CASP1 P29466 1/20 0.56
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CYP1A2 P05177 1/20 0.48
PDGFRB P09619 2/20 0.47
PDGFRA P16234 2/20 0.47
CYP2A6 P11509 1/20 0.45
NISCH Q9Y2I1 1/20 0.44
MGAM O43451 1/20 0.43
HTR3A P46098 1/20 0.43
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14678 0.90 CYP1A2 (0.57) ALDH1A1HSP90AA1MAPTATMKDM4E
SCHEMBL29418017 0.90 CYP1A2 (0.57) ALDH1A1HSP90AA1MAPTATMKDM4E
Quinoline SCHEMBL28292612 0.89 ALDH1A1 (0.67) ALDH1A1HSP90AA1MAPTATMKDM4E
Hydrochloric Acid SCHEMBL29862578 0.88 CYP1A2 (0.55) ALDH1A1HSP90AA1MAPTATMKDM4E
Hydrochloric Acid SCHEMBL8324913 0.88 CYP1A2 (0.55) ALDH1A1HSP90AA1MAPTATMKDM4E
Hydrochloric Acid SCHEMBL7362443 0.88 CYP1A2 (0.55) ALDH1A1HSP90AA1MAPTATMKDM4E
Ethylene SCHEMBL28325267 0.86 CYP1A2 (0.53) ALDH1A1HSP90AA1MAPTATMKDM4E
Acetic Acid SCHEMBL7836636 0.79 MGAM (0.57) ALDH1A1HSP90AA1MAPTATMKDM4E
SCHEMBL4944778 0.76 KMT2A (0.44) ALDH1A1HSP90AA1MAPTATMKDM4E
SCHEMBL29818168 0.76 PDGFRB (0.62) CYP1A2PDGFRBPDGFRACYP2A6NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2142503-A2 PROCESS FOR THE MANUFACTURE FOR NON-STEROIDAL ANTI-INFLAMMATORY AGENTS AND INTERMEDIATES THEREOF Intendis GmbH (DE) 2010-01-13 EP claimed
WO-2008128750-A2 PROCESS FOR THE MANUFACTURE FOR NON-STEROIDAL ANTI-INFLAMMATORY AGENTS AND INTERMEDIATES THEREOF INTENDIS GMBH (DE) 2008-10-30 WO claimed
EP-2142503-A2 PROCESS FOR THE MANUFACTURE FOR NON-STEROIDAL ANTI-INFLAMMATORY AGENTS AND INTERMEDIATES THEREOF Intendis GmbH (DE) 2010-01-13 EP disclosed
WO-2008128750-A2 PROCESS FOR THE MANUFACTURE FOR NON-STEROIDAL ANTI-INFLAMMATORY AGENTS AND INTERMEDIATES THEREOF INTENDIS GMBH (DE) 2008-10-30 WO disclosed