SCHEMBL28537113

SCHEMBL28537113

CC(=O)Nc1ccc(C2=CCN(C(=O)O)CC2)cc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.46
NPSR1 Q6W5P4 1/20 0.46
QDPR P09417 2/20 0.46
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 2/20 0.42
HTT P42858 2/20 0.42
ALDH1A1 P00352 7/20 0.41
NPC1 O15118 2/20 0.41
ALOX15 P16050 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 1/20 0.41
HPGD P15428 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
ABCB1 P08183 2/20 0.39
ABCC1 P33527 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28551485 0.92 QDPR (0.55) MAPTNPSR1QDPRPOLBPKM
SCHEMBL28543598 0.86 NAMPT (0.52) MAPTNPSR1QDPRKMT2A
SCHEMBL28614009 0.84 KMT2A (0.47) MAPTNPSR1POLBPKMKMT2A
SCHEMBL27037449 0.82 QDPR (0.54) MAPTQDPRKMT2AALDH1A1NPC1
SCHEMBL17398277 0.81 QDPR (0.47) QDPRKMT2AHTTALDH1A1NPC1
SCHEMBL3986410 0.81 QDPR (0.44) MAPTNPSR1QDPRKMT2AHTT
SCHEMBL3986414 0.81 QDPR (0.44) MAPTNPSR1QDPRKMT2AHTT
SCHEMBL16262930 0.81 MAPT (0.50) MAPTNPSR1QDPRPOLBKMT2A
SCHEMBL17398284 0.81 QDPR (0.47) QDPRKMT2AHTTALDH1A1NPC1
SCHEMBL16262927 0.81 MAPT (0.50) MAPTNPSR1QDPRPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107400092-B Pyrimidine derivative, preparation method thereof and application thereof in medicine 浙江海正药业股份有限公司 2021-08-24 CN disclosed
CN-108264511-B Heterocyclic derivative, preparation method thereof and application thereof in medicine 浙江海正药业股份有限公司 2021-04-13 CN disclosed