SCHEMBL28537305

SCHEMBL28537305

CC(C)(C)c1nc(Cl)nc(NC2CCC2)c1C#N

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
HPGD P15428 4/20 0.40
GAA P10253 3/20 0.40
HSD17B10 Q99714 1/20 0.40
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
HIF1A Q16665 1/20 0.37
PDE4A P27815 2/20 0.36
ACHE P22303 2/20 0.36
NPSR1 Q6W5P4 2/20 0.35
PDE10A Q9Y233 1/20 0.34
CTSK P43235 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34
ULK1 O75385 1/20 0.33
AXL P30530 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30042311 0.67 KMT2A (0.56) ALDH1A1KMT2AACHECTSKULK1
SCHEMBL21596374 0.67 KMT2A (0.56) ALDH1A1KMT2AACHECTSKULK1
SCHEMBL11169614 0.66 PDE4A (0.44) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL13165484 0.65 PDE10A (0.36) KMT2APDE4APDE10AADORA3ADORA1
SCHEMBL4416389 0.64 ACHE (0.43) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL11174566 0.64 HTT (0.41) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL16714483 0.63 KMT2A (0.44) KMT2APDE4APDE10ACTSKADORA3
SCHEMBL2816729 0.63 KMT2A (0.62) ALDH1A1KMT2AACHECTSKAXL
SCHEMBL22430981 0.62 CHUK (0.43) KMT2AADORA3ADORA1AXL
SCHEMBL15589491 0.62 PDE4A (0.54) KMT2APDE4APDE10AAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112313207-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-02-02 CN disclosed