SCHEMBL28538511

SCHEMBL28538511

Cn1c(=O)c2c(ncn2CCOc2ccc(/C=C/C(=O)O)cc2)n(C)c1=O

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 6/20 0.67
ADORA2B P29275 4/20 0.57
LMNA P02545 1/20 0.52
TBXAS1 P24557 2/20 0.52
PDE3A Q14432 2/20 0.51
ADORA1 P30542 1/20 0.51
ALDH1A1 P00352 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KMT2A Q03164 1/20 0.49
MAPK1 P28482 1/20 0.49
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30810227 1.00 RXFP1 (0.67) RXFP1ADORA2BLMNATBXAS1PDE3A
SCHEMBL28547018 0.84 RXFP1 (0.74) RXFP1ADORA2BLMNAPDE3AALDH1A1
SCHEMBL28551846 0.82 ADORA2B (0.58) RXFP1ADORA2BLMNATBXAS1PDE3A
SCHEMBL30810148 0.82 ADORA2B (0.58) RXFP1ADORA2BLMNATBXAS1PDE3A
SCHEMBL30810165 0.80 KDM4E (0.54) RXFP1ADORA2BALDH1A1SMN1; SMN2MAPK1
SCHEMBL28557871 0.80 KDM4E (0.54) RXFP1ADORA2BALDH1A1SMN1; SMN2MAPK1
SCHEMBL7141074 0.78 RXFP1 (0.73) RXFP1ADORA2BLMNAPDE3AALDH1A1
SCHEMBL11380427 0.76 RXFP1 (0.55) RXFP1ADORA2BLMNAALDH1A1SMN1; SMN2
SCHEMBL11380423 0.76 RXFP1 (0.55) RXFP1ADORA2BLMNAALDH1A1SMN1; SMN2
SCHEMBL11382728 0.74 ADORA2B (0.56) RXFP1ADORA2BLMNAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112500413-B Xanthine aromatic acid ether derivatives, preparation method and application thereof 安徽中医药大学 2024-03-01 CN disclosed
CN-112500413-A Xanthine aromatic acid ether derivatives and application thereof 安徽中医药大学 2021-03-16 CN disclosed