SCHEMBL28547018

SCHEMBL28547018

Cn1c(=O)c2c(ncn2CCOc2ccc(C(=O)O)cc2)n(C)c1=O

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 6/20 0.74
ADORA2B P29275 7/20 0.63
PDE3A Q14432 2/20 0.58
LMNA P02545 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.55
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.54
MAPK1 P28482 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28538511 0.84 RXFP1 (0.67) RXFP1ADORA2BPDE3ALMNASMN1; SMN2
SCHEMBL30810227 0.84 RXFP1 (0.67) RXFP1ADORA2BPDE3ALMNASMN1; SMN2
SCHEMBL28547032 0.83 RXFP1 (0.60) RXFP1ADORA2BLMNASMN1; SMN2ALDH1A1
SCHEMBL7141074 0.83 RXFP1 (0.73) RXFP1ADORA2BPDE3ALMNASMN1; SMN2
SCHEMBL29256880 0.82 ADORA2B (0.74) RXFP1ADORA2BLMNASMN1; SMN2ALDH1A1
SCHEMBL28543990 0.81 ADORA2B (0.64) RXFP1ADORA2BPDE3ALMNASMN1; SMN2
SCHEMBL10966452 0.80 RXFP1 (0.64) RXFP1ADORA2BSMN1; SMN2ALDH1A1
SCHEMBL30810226 0.80 ADORA2B (0.61) RXFP1ADORA2BLMNASMN1; SMN2ALDH1A1
SCHEMBL28025751 0.78 ADORA2B (1.00) RXFP1ADORA2BLMNASMN1; SMN2MAPT
SCHEMBL28547575 0.78 CYP1A2 (0.54) RXFP1ADORA2BPDE3ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112500413-B Xanthine aromatic acid ether derivatives, preparation method and application thereof 安徽中医药大学 2024-03-01 CN disclosed
CN-112500413-A Xanthine aromatic acid ether derivatives and application thereof 安徽中医药大学 2021-03-16 CN disclosed