SCHEMBL28539140

SCHEMBL28539140

CC(=O)c1c(C)[nH]c(-c2nc3ccccc3[nH]2)c1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 18/20 1.00
SMN1; SMN2 Q16637 1/20 0.56
AURKA O14965 1/20 0.50
CDK1 P06493 1/20 0.50
CCNB1 P14635 1/20 0.50
CDK2 P24941 1/20 0.50
AURKB Q96GD4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28451053 0.84 BRD4 (0.73) BRD4SMN1; SMN2
SCHEMBL30532574 0.84 BRD4 (0.73) BRD4SMN1; SMN2
SCHEMBL28539261 0.81 BRD4 (0.77) BRD4
SCHEMBL28544075 0.79 BRD4 (0.65) BRD4SMN1; SMN2
SCHEMBL28911157 0.79 BRD4 (0.65) BRD4SMN1; SMN2
SCHEMBL28539642 0.79 BRD4 (0.65) BRD4
SCHEMBL28546032 0.78 BRD4 (1.00) BRD4SMN1; SMN2
SCHEMBL28546029 0.78 BRD4 (1.00) BRD4
SCHEMBL1799622 0.73 ALDH1A1 (0.60) BRD4SMN1; SMN2
SCHEMBL1799620 0.73 BRD4 (0.57) BRD4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107739370-B Preparation method and application of pyrrolidone BRD4 protein inhibitor 中国药科大学 2021-03-30 CN claimed
CN-107739370-B Preparation method and application of pyrrolidone BRD4 protein inhibitor 中国药科大学 2021-03-30 CN disclosed