SCHEMBL28539261

SCHEMBL28539261

CC(=O)c1c(C)[nH]c(-c2nc3ccc(C(=O)O)cc3[nH]2)c1C

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 15/20 0.77
HSP90AA1 P07900 1/20 0.56
ESR2 Q92731 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
NR4A2 P43354 1/20 0.52
CHEK2 O96017 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28546032 0.87 BRD4 (1.00) BRD4
SCHEMBL1799622 0.82 ALDH1A1 (0.60) BRD4CHEK2
SCHEMBL28910531 0.82 BRD4 (0.72) BRD4
SCHEMBL28539642 0.81 BRD4 (0.65) BRD4
SCHEMBL28539143 0.81 BRD4 (0.74) BRD4
SCHEMBL28539140 0.81 BRD4 (1.00) BRD4
SCHEMBL28546029 0.80 BRD4 (1.00) BRD4
SCHEMBL28547542 0.78 BRD4 (1.00) BRD4
SCHEMBL28542913 0.77 BRD4 (1.00) BRD4
SCHEMBL1802494 0.75 BRD4 (0.59) BRD4CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107739370-B Preparation method and application of pyrrolidone BRD4 protein inhibitor 中国药科大学 2021-03-30 CN disclosed