SCHEMBL28539313

SCHEMBL28539313

Cc1cc2cc(Br)ccc2nc1-c1ccc(Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.53
BACE1 P56817 1/20 0.43
PRNP P04156 1/20 0.43
AURKA O14965 2/20 0.43
AURKB Q96GD4 2/20 0.43
KDR P35968 1/20 0.43
MAPT P10636 4/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
AKR1B10 O60218 1/20 0.40
DHODH Q02127 3/20 0.40
PSMB5 P28074 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
APP P05067 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28536639 0.89 PDE10A (0.69) PDE10APRNPAURKBMAPTALDH1A1
SCHEMBL28853907 0.86 PDE10A (0.74) PDE10APRNPMAPTALDH1A1TDP1
SCHEMBL8733061 0.85 DHODH (0.53) PDE10AAKR1B10DHODH
SCHEMBL12578166 0.79 MAPK14 (0.56) PDE10AAURKAAURKBMAPTALDH1A1
SCHEMBL11872346 0.79 TDP1 (0.62) PDE10ABACE1ALDH1A1HTTPSMB5
SCHEMBL4143806 0.77 PDE10A (0.56) PDE10ABACE1MAPTALDH1A1MAPK1
SCHEMBL1128599 0.76 BACE1 (0.44) BACE1MAPTALDH1A1HTTSMN1; SMN2
SCHEMBL789778 0.76 BACE1 (0.53) BACE1MAPTALDH1A1HTTPSMB5
SCHEMBL12317094 0.74 ALDH1A1 (0.68) AURKAAURKBKDRMAPTALDH1A1
SCHEMBL22804126 0.74 NPC1 (0.39) PDE10AMAPTALDH1A1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112521333-A Synthesis method of chiral 2, 3-disubstituted tetrahydroquinoline derivative 中国科学院大连化学物理研究所 2021-03-19 CN disclosed