SCHEMBL28539714

SCHEMBL28539714

COCCOc1ccc2c(c1)CCN(C(=O)O)C2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
HRH3 Q9Y5N1 6/20 0.51
SCN9A Q15858 1/20 0.48
KMT2A Q03164 2/20 0.48
ABHD6 Q9BV23 2/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
TAAR1 Q96RJ0 1/20 0.45
PPARG P37231 3/20 0.45
PPARD Q03181 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28533346 0.95 HRH3 (0.57) ESR1ESR2HRH3SCN9AKMT2A
SCHEMBL21659712 0.84 ESR2 (0.63) ESR1ESR2HRH3SCN9AKMT2A
SCHEMBL11295872 0.84 ESR1 (0.71) ESR1ESR2KMT2AABHD6HPGD
SCHEMBL5137232 0.83 HRH3 (0.58) HRH3KMT2AABHD6HPGDTSHR
SCHEMBL30290475 0.83 HRH3 (0.52) ESR1ESR2HRH3KMT2AABHD6
SCHEMBL21659498 0.80 NR1H2 (0.62) ESR1ESR2HRH3KMT2AABHD6
SCHEMBL23701210 0.79 HRH3 (0.49) ESR1ESR2HRH3KMT2AABHD6
SCHEMBL29168677 0.79 DRD1 (0.40) ESR1ESR2HRH3KMT2AHPGD
SCHEMBL27538580 0.78 HRH3 (0.52) ESR1ESR2HRH3KMT2AHPGD
SCHEMBL29168624 0.77 HSP90AA1 (0.38) ESR1ESR2HRH3SCN9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112469722-A Pyrazolo-triazolopyrimidine derivatives as A2A receptor antagonists 百济神州有限公司 2021-03-09 CN disclosed