SCHEMBL28539729

SCHEMBL28539729

S=C(NCc1cccc2ccccc12)Nc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.68
MEN1 O00255 2/20 0.68
KMT2A Q03164 2/20 0.68
MAOB P27338 3/20 0.63
MAOA P21397 1/20 0.63
ALOX12 P18054 2/20 0.55
HPGD P15428 2/20 0.55
CA9 Q16790 1/20 0.55
ALDH1A1 P00352 2/20 0.54
PPARG P37231 1/20 0.54
NCOA3 Q9Y6Q9 1/20 0.54
POLB P06746 1/20 0.53
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
NPSR1 Q6W5P4 1/20 0.51
LMNA P02545 1/20 0.51
PLA2G1B P04054 1/20 0.51
ATG4B Q9Y4P1 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28912557 0.81 MEN1 (1.00) MAPTMEN1KMT2AMAOBHPGD
SCHEMBL13779437 0.81 ALOX12 (0.54) MAPTMEN1KMT2AALOX12HPGD
SCHEMBL13779436 0.81 MTNR1A (0.51) MAPTMEN1KMT2A
SCHEMBL5452784 0.79 KMT2A (0.63) MAPTMEN1KMT2AALDH1A1POLB
SCHEMBL1520659 0.78 MAOB (1.00) MAPTMEN1KMT2AMAOBMAOA
SCHEMBL31674408 0.78 MAOB (0.62) MAPTMEN1KMT2AMAOBMAOA
SCHEMBL5524250 0.77 MTNR1A (0.57) MAPTMEN1KMT2AHPGD
SCHEMBL30388749 0.77 MAOB (0.83) MAPTMEN1KMT2AMAOBMAOA
SCHEMBL30849357 0.76 MAPT (0.49) MAPTMEN1KMT2AMAOBMAOA
SCHEMBL29207165 0.76 MAPT (0.49) MAPTMEN1KMT2AMAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574082-B Preparation method of thiourea alkylated derivative 西华大学 2022-07-29 CN disclosed
CN-112574082-A Preparation method of thiourea alkylated derivative 西华大学 2021-03-30 CN disclosed